Sociedad Americana de Hirudoterapia

Pharmacology of recombinant hirudin

Research article published in Seminars in thrombosis and hemostasis (2002)

Última actualización: March 18, 2026Revisado por: ASH Editorial Board
Research article — evidence reviewArticle reference
Desarrollo de fármacosFarmacología salivalGenómica y proteómicaNowak G · Seminars in thrombosis and hemostasis, 2002

Abstract

Hirudin is the anticoagulative product of the salivary glands of the medical leech Hirudo medicinalis. It is characterized by a direct, bifunctional inhibition mechanism and a high, exclusive specificity and a strong ability to bind to thrombin (tight binding). Further characteristics are the organic-chemical structure of hirudin (peptide), which allows only parenteral administration; the missing metabolism in the organism; and the exclusive glomerular filtration of hirudin in kidneys as the effective elimination mechanism. Recombinant hirudin (r-hirudin) is a product of genetic engineering that is identical to the hirudin found in nature and has the same biochemical and pharmacological characteristics as natural hirudin.

Abstract sourced from PubMed (NCBI) for the cited record. See the original publication for the authoritative version.

Publication typeJournal ArticleReview
Indexed MeSH termsAmino Acid SequenceAnimalsDose-Response Relationship, DrugFibrinolytic AgentsGenetic EngineeringHirudin TherapyHirudinsHumansLeechesMolecular Sequence DataProtein Structure, SecondaryProtein Structure, Tertiary

Resumen

Hirudin is the anticoagulative product of the salivary glands of the medical leech Hirudo medicinalis. It is characterized by a direct, bifunctional inhibition mechanism and a high, exclusive specificity and a strong ability to bind to thrombin (tight binding).

Por qué esto importa para la hirudoterapia

Relevant to the development and clinical application of leech-derived pharmaceutical compounds.

Citación

Pharmacology of recombinant hirudin.

Nowak G · Seminars in thrombosis and hemostasis, 2002

Contexto clínico relacionado

Añadido a la biblioteca ASH: March 18, 2026 · Última actualización del sitio: March 18, 2026

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Pharmacology of recombinant hirudin | ASH